ISSN 1004-6879

CN 13-1154/R

 

承德医学院学报 ›› 2018, Vol. 35 ›› Issue (1): 11-14.

• 基础医学 • 上一篇    下一篇

秦皮乙素降低多柔比星诱导心脏毒性的研究*

李潇, 徐繁, 房亮, 曹向宇, 姜海军, 肖旭   

  1. 承德医学院附属医院,河北承德 067000
  • 收稿日期:2017-04-04 出版日期:2018-02-10 发布日期:2021-11-21
  • 通讯作者:
  • 基金资助:
    * 河北省2017年度医学科学研究重点课题计划(20170886)

STUDY ON ESCULETIN REDUCE CARDIOTOXICITY INDUCED BY DOXORUBICIN

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  1. the Affiliated Hospital of Chengde Medical College, Hebei Chengde 067000, China
  • Received:2017-04-04 Online:2018-02-10 Published:2021-11-21

摘要: 目的: 探讨秦皮乙素(Esc)对多柔比星(DOX)诱导的H9C2细胞损伤的保护作用及机制。方法: 培养H9C2心肌细胞并分为对照组、模型(DOX)组和干预(Esc+DOX)组。流式细胞术检测细胞凋亡情况和细胞内活性氧(ROS)的水平;蛋白印迹法检测cleaved Caspase-3、cleaved PARP、Bid和Bcl-2蛋白的表达情况。结果: 模型组H9C2细胞凋亡数量、ROS水平,cleaved Caspase-3、cleaved PARP、Bid蛋白表达明显高于对照组,Bcl-2蛋白表达明显低于对照组(P<0.05);干预组H9C2细胞凋亡数量、ROS水平,cleaved Caspase-3、cleaved PARP、Bid蛋白表达明显低于模型组,Bcl-2蛋白表达明显高于模型组(P<0.05)。结论: 秦皮乙素可减轻多柔比星所致的心脏毒性,其作用机制与减少细胞凋亡、降低ROS水平有关。

关键词: 多柔比星, 秦皮乙素, 心脏毒性

Abstract: Objective: To investigate the protective effects and mechanisms of esculetin (Esc) on H9C2 cells injury induced by doxorubicin (DOX). Methods: The H9C2 cells were cultured and divided into control group, model (DOX) group and intervention (Esc+DOX) group. Flow cytometry was used to detect apoptosis of H9C2 cells and reactive oxygen (ROS) level in H9C2 cells; Western blotting to detect the cleaved Caspase-3, cleaved PARP, Bid and Bcl-2 protein expression in H9C2 cells. Results: The number of apoptosis, ROS level, cleaved Caspase-3, cleaved PARP and Bid protein expression in H9C2 cells in model group were obviously higher than control group; the Bcl-2 protein expression were obviously lower (P<0.05). The number of apoptosis, ROS level, cleaved Caspase-3, cleaved PARP and Bid protein expression in H9C2 cells in intervention group were obviously lower than model group; the Bcl-2 protein expression were obviously higher (P<0.05). Conclusions: Esculetin can reduce cardiotoxicity induced by doxorubicin by reducing apoptosis and ROS level.

Key words: Doxorubicin, Esculetin, Cardiotoxicity

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